Browsing by Author "Moreira, Diogo Rodrigo Magalhães"
Now showing items 37-54 of 54
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Phthalimido-thiazoles as building blocks and their effects on the growth and morphology of Trypanosoma cruzi.
Gomes, Paulo André Teixeira de Moraes et al. | Date Issued: 2016 -
Physalins B and F, seco-steroids isolated from Physalis angulata L., strongly inhibit proliferation, ultrastructure and infectivity of Trypanosoma cruzi.
Meira, Cássio Santana et al. | Date Issued: 2013 -
Potencial citotóxico de novos complexos de rutênio contendo piplartina como ligante
Costa, Cinara Oliveira D'Sousa | Date Issued: 2017INTRODUÇÃO: A quimioterapia ainda é uma importante forma de tratamento de diversos tipos de cânceres; entretanto, as células cancerosas podem adquirirem resistência aos agentes quimioterápicos, que por sua vez, também induzem ... -
Potent immunosuppressive activity of a phosphodiesterase-4 inhibitor N-acylhydrazone in models of lipopolysaccharide-induced shock and delayed-type hypersensitivity reaction
Guimarães, Elisalva Teixeira et al. | Date Issued: 2018 -
Ruthenium complexes endowed with potent anti-Trypanosoma cruzi activity: Synthesis, biological characterization and structure-activity relationships
Donnici, Claudio Luis et al. | Date Issued: 2009 -
Ruthenium(II) complexes of 1,3-thiazolidine-2-thione: Cytotoxicity against tumor cells and anti-Trypanosoma cruzi activity enhanced upon combination with benznidazole.
Corrêa, Rodrigo S et al. | Date Issued: 2016 -
Structural design, synthesis and pharmacological evaluation of 4-thiazolidinones against Trypanosoma cruzi
Oliveira Filho, Gevanio Bezerra de et al. | Date Issued: 2015 -
Structural design, synthesis and structure-activity relationships of thiazolidinones with enhanced anti-Trypanosoma cruzi activity
Moreira, Diogo Rodrigo Magalhães et al. | Date Issued: 2014 -
Structural Insights Into Bioactive Thiazolidin-4-one: Experimental and Theoretical Data
Cardoso, Marcos Veríssimo de Oliveira et al. | Date Issued: 2015Although viewed as promising drug candidates, few efforts have been addressed towards the structural chemistry of 2-hydrazonothiazolidin-4-ones. Therefore, 2-[(3-phenylsulfanylpropylidene)- hydrazono]thiazolidin-4-one ... -
Structural investigation of anti-Trypanosoma cruzi 2-iminothiazolidin-4-ones allows the identification of agents with efficacy in infected mice.
Moreira, Diogo Rodrigo Magalhães et al. | Date Issued: 2012 -
Structural planning, synthesis and evaluation of properties trypanocidal aryl-1,3-thiazoles
Barbosa, Miria de Oliveira et al. | Date Issued: 2016 -
Structure-activity relationships of mononuclear metal-thiosemicarbazone complexes endowed with potent antiplasmodial and antiamoebic activities.
Bahl, Deepa et al. | Date Issued: 2010 -
Synthesis and structure-activity relationship study of a new series of antiparasitic aryloxyl thiosemicarbazones inhibiting Trypanosoma cruzi cruzain.
Espíndola, José Wanderlan Pontes et al. | Date Issued: 2015 -
Synthesis of 4'-(2-ferrocenyl)-2,2':6'2''-terpyridine: characterization and antiprotozoal activity of Mn(II), Co(II), Ni(II), Cu(II) and Zn(II) complexes.
Juneja, Annu et al. | Date Issued: 2014 -
Synthesis of piplartine analogs and preliminary findings on structure–antimicrobial activity relationship
Fregnan, Antonio Maciel et al. | Date Issued: 2017 -
Synthesis, Cruzain docking, and in vitro studies of aryl-4-oxothiazolylhydrazones against Trypanosoma cruzi.
Leite, Ana Cristina Lima et al. | Date Issued: 2007 -
Synthesis, docking, and in vitro activity of thiosemicarbazones, aminoacyl-thiosemicarbazides and acyl-thiazolidones against Trypanosoma cruzi
Leite, Ana Cristina Lima et al. | Date Issued: 2006 -
Synthesis, in vitro and in vivo biological evaluation, COX-1/2 inhibition and molecular docking study of indole-N-acylhydrazone derivatives
Moraes, Ana Daura Travassos de Oliveira et al. | Date Issued: 2018